ClinPharm Vault
A Study of GDC-0853 in Participants With Refractory Chronic Spontaneous Urticaria (CSU).
Study Snapshot
- Program: Fenebrutinib
- Study ID(s): NCT03137069
- Phase: Phase 2
- Indication: Urticaria
- Status: Completed
- Sponsor: Genentech, Inc.
Design
- Study type: INTERVENTIONAL
- Randomization / allocation: RANDOMIZED
- Intervention model: PARALLEL
- Masking: QUADRUPLE
- Primary purpose: TREATMENT
- Enrollment: 134 (ACTUAL)
Population
- Conditions: Urticaria
- Sex: ALL
- Age range: 18 Years to 75 Years
- Healthy volunteers: False
- Summary: The purpose of this study is to evaluate the efficacy, safety and pharmacokinetics of GDC-0853 compared with placebo in participants with Refractory Chronic Spontaneous Urticaria (CSU) already treated with anti-histamines. Participants have the option to enter the Open-Label Extension (OLE) study after completing the 8-week treatment period.
Operational design summary
- Arms represented in current CT.gov export: 6
- Active dose regimens represented in current local source layer: 3
- Total study enrollment in CT.gov: 134 (ACTUAL)
- Design interpretation: Pilot plus dose-ranging fenebrutinib phase 2 study with separate cohort 1 and cohort 2 structures.
- Per-arm sample size summary: ClinicalTrials.gov results-section denominators support cohort 1 placebo n=13 and fenebrutinib 200 mg BID n=28, plus cohort 2 placebo n=23, fenebrutinib 50 mg daily n=23, 150 mg daily n=24, and 200 mg twice daily n=23, totaling 134 participants.
- Arm-size evidence source: ClinicalTrials.gov API v2 resultsSection participant flow and baseline-characteristics denominators; PMCID PMC8604722 full text remains the linked manuscript source.
Arms
| Arm | Type | Dose | Frequency | Route | Description | N | Evidence status |
|---|---|---|---|---|---|---|---|
| Cohort 1: Placebo | PLACEBO_COMPARATOR | NR | BID | NR | Participants received matching placebo twice daily from Day 1 to 56. | 13 | Directly supported by linked local publication/source text or explicit CT.gov arm-level enrollment context |
| Cohort 1: GDC-0853 200mg BID | EXPERIMENTAL | 200mg | BID | NR | Participants received GDC-0853 200mg twice daily from Day 1 to 56. | 28 | Directly supported by linked local publication/source text or explicit CT.gov arm-level enrollment context |
| Cohort 2: Placebo | PLACEBO_COMPARATOR | NR | BID | NR | Participants received matching placebo up to twice daily from Day 1 to 56. | 23 | Directly supported by linked local publication/source text or explicit CT.gov arm-level enrollment context |
| Cohort 2: GDC-0853 50mg QD | EXPERIMENTAL | 50mg | QD | NR | Participants received GDC-0853 50mg once daily from Day 1 to 56. | 23 | Directly supported by linked local publication/source text or explicit CT.gov arm-level enrollment context |
| Cohort 2: GDC-0853 150mg QD | EXPERIMENTAL | 150mg | QD | NR | Participants received GDC-0853 150mg once daily from Day 1 to 56. | 24 | Directly supported by linked local publication/source text or explicit CT.gov arm-level enrollment context |
| Cohort 2: GDC-0853 200mg BID | EXPERIMENTAL | 200mg | BID | NR | Participants received GDC-0853 200mg twice daily from Day 1 to 56. | 23 | Directly supported by linked local publication/source text or explicit CT.gov arm-level enrollment context |
Key Efficacy and Safety Findings
- Result status: Published
Efficacy
- Cohort 2 primary endpoint (UAS7 change at week 8, LS mean difference versus placebo): 200 mg BID -9.5 (95% CI -16.7 to -2.4; significant), 150 mg QD -6.4 (95% CI -13.4 to 0.6; trend), 50 mg QD -0.5 (not significant).
- Well-controlled disease (UAS7 <= 6) at week 8: 200 mg BID 57%, 150 mg 46%, 50 mg 35%, placebo 22%.
- Complete response (UAS7 = 0) at week 8: 200 mg BID 39%, 150 mg 25%, 50 mg 13%, placebo 4%.
- Rapid onset: 200 mg BID week-4 UAS7 LS mean difference -10.8 versus placebo (95% CI -18.2 to -3.3).
- Exploratory: all doses reduced IgG-anti-FcεRI autoantibodies (median change -43.7% to -53.6% versus +20.4% placebo).
Safety
- No SAEs in Cohort 2; most common AEs: urticaria (15%), nasopharyngitis (11%), headache (6%).
- Grade 2/3 liver transaminase elevations in 2 patients each at 150 mg QD and 200 mg BID; all asymptomatic and reversible.
- Dose-dependent creatinine increases starting week 1; no serious or opportunistic infections.
- Note: further CSU studies of fenebrutinib are not planned; program pivoted to MS.
Result source(s)
- PMID 34750553
- PMCID PMC8604722
Endpoints
- Primary outcomes:
- Change From Baseline in the Urticaria Activity Score Over 7 Days (UAS7) at Day 57 (time frame: Baseline and Day 57)
Clinical Pharmacology Findings
- PK: ClinicalTrials.gov summary text indicates pharmacokinetics were part of the study objectives or assessments.
- PD: Not clearly summarized in the currently linked local source snippets.
- Linked manuscripts: No trial-level primary publication is explicitly linked in the current registry.
Safety Findings
- Safety detail is not strongly enriched beyond the current CT.gov/source-registry layer.
Linked Evidence
- CT.gov page: https://clinicaltrials.gov/study/NCT03137069
- Local CT.gov cache:
raw/clinicaltrials/markdown/NCT03137069.md
Interpretation
- Verified facts: this page reflects the current local registry and CT.gov inventory export without inferring unsupported arm sizes or endpoint results.
- Interpretation: this trial is currently represented mainly by CT.gov and any linked sponsor-source artifacts; manual enrichment is still needed for a richer narrative page.
- Open questions:
- Some studies still lack exact arm-specific N in the current promoted evidence layer even when allocation schema or total enrollment is visible.
- No explicit trial-level primary manuscript is currently linked in the registry.
- No sponsor artifact is explicitly linked to this trial by identifier in the current registry.
Provenance
- Source type: ClinicalTrials.gov inventory with linked sponsor/publication registry where available
- Primary source(s):
- NCT03137069
../raw/clinicaltrials/markdown/NCT03137069.md../inventories/source_registry.json- Supporting source(s):
../inventories/ctgov_priority_trials.json- Last verified: 2026-04-08
- Verification status: Partial
Change Log
- 2026-04-08: Generated or refreshed this study page from the v2 source registry and CT.gov inventory.